Teko e Ncha ea Kliniki bakeng sa Kalafo ea Kankere ea tšoelesa ea senya

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Avatar ea Linda Hohnholz
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Hinova Pharmaceuticals Inc., k'hamphani ea bongaka ea biopharmaceutical e tsepamisitseng maikutlo ho nts'etsopele ea kalafo e ncha bakeng sa mofets'e le mafu a metabolic ka theknoloji e shebiloeng ea ho senyeha ha protheine, e phatlalalitse hore mokuli oa pele ea nang le mofetše oa tšoelesa ea senya ea metastatic castration-resistant prostate (mCRPC) o atlehile ho fuoa litekanyetso Mokhahlelong oa I. teko ea tleliniki ea HP518, e khethollang haholo le ka molomo bioavailable chimeric degrader targeting androgen receptor (AR). Boithuto bo tsoelang pele ba li-label Phase I ho la Australia bo tla lekola polokeho, pharmacokinetics, le ts'ebetso ea anti-tumor ea HP518 ho bakuli ba nang le mCRPC.

HP518 e sibollotsoe le ho ntlafatsoa ke sethala sa Hinova sa ho sibolla lithethefatsi tse senyang protheine. E na le monyetla oa ho hlola khanyetso ea lithethefatsi ea mofetše oa senya ka lebaka la liphetoho tse itseng tsa AR.

Li-degraders tsa Chimeric ke limolek'hule tse nyenyane tse sebetsang habeli tse khothalletsang ho senyeha ha liprotheine tse lebisitsoeng tse nang le matla a phahameng le khetho e phahameng. Theknoloji ena e na le monyetla oa ho shebana le lipheo tse sa sebeliseng lithethefatsi le ho hlola taba ea khanyetso ea lithethefatsi ea litlhare tse tloaelehileng tsa molek'hule.

"Ena ke ketsahalo ea bohlokoa tsoelo-peleng ea boiteko ba rona ho tloha ho sibollo ea lithethefatsi ho fihlela thutong ea bongaka," ho boletse Yuanwei Chen, Ph.D., Mopresidente le CEO oa Hinova. "Re thabile ka hona 'me re ikemiselitse ho tlisa mekhoa e mecha ea phekolo ho bakuli lefatšeng ka bophara!"

Ka sethala se reriloeng sa ho sibolla lithethefatsi tsa protheine, Hinova e khona ho shebisisa ts'ebetso ea pholiso ea protheine kapele mme e fihlelle moralo o nepahetseng le ntlafatso ea li-chimeric degraders. Ho feta moo, Hinova o na le phihlelo e tebileng ea ho laola lik'hemik'hale tsa lik'hemik'hale tsa Chimeric degrader compounds.

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Avatar ea Linda Hohnholz

Linda Hohnholz

Mohlophisi e ka sehloohong bakeng sa eTurboNews e thehiloe ho eTN HQ.

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